Chemistry: DD3 Modern Tactics to Optimise Potency Updated
Description
When you have 1000s of possible compounds you could make from any one start point what do you make first? This lecture will cover some general basic principles on designing more potent molecules, as well as some practical tips on how to run an optimization program and how to focus synthetic efforts. Binding modalities (reversible, covalent) will be briefly covered, as well as some newer non-traditional modalities. This lecture will also serve as an introduction to the medicinal chemistry game.
Target audience
- Chemistry postgraduates
- Further details regarding eligibility criteria are available
Duration
- One session of one hour
Theme
Drug Discovery
Events available